Summary

Top ## selected# in Chembl# in DrugBank# in Kegg# in any DB
100 (0%)0 (0%)0 (0%)0 (0%)0 (0%)
200 (0%)0 (0%)0 (0%)0 (0%)0 (0%)
500 (0%)0 (0%)0 (0%)0 (0%)0 (0%)
1001 (1%)0 (0%)0 (0%)0 (0%)0 (0%)
2009 (4%)1 (11%)0 (0%)1 (11%)2 (22%)
50089 (18%)4 (4%)5 (6%)3 (3%)10 (11%)
1000332 (33%)17 (5%)18 (5%)7 (2%)37 (11%)

Ranking of Drug—Target Pairs

Rank CH DB KG Drug Target Most Similar Drug Most Similar Target
61NNNEletriptan hydrobromide
HTR6: 5-hydroxytryptamine (serotonin) receptor 60.42857Olanzapine
0.21266HTR7: 5-hydroxytryptamine (serotonin) receptor 7 (adenylate cyclase-coupled)
101NNNCinnarizine
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.44118Mianserin hydrochloride
0.18620DRD3: dopamine receptor D3
117NNNPindolol
DRD4: dopamine receptor D40.31250Propiomazine
0.24654ADRA2A: alpha-2A adrenergic receptor
140NNNTamsulosin hydrochloride
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.48485Promethazine
0.18839ADRA1B: alpha-1B adrenergic receptor
173YNNSumatriptan
DRD2: dopamine receptor D20.41379Chlorpromazine
0.24883HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
176NNNOlanzapine
HRH3: histamine receptor H30.40000Astemizole
0.24459CHRM1: cholinergic receptor, muscarinic 1
182NNYEnprostil
PTGER2: prostaglandin E receptor 2 (subtype EP2), 53kDa0.47368Misoprostol
0.16952PTGER3: prostaglandin E receptor 3 (subtype EP3)
194NNNPindolol
CHRM1: cholinergic receptor, muscarinic 10.35714Promethazine
0.21367HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
197NNNEletriptan hydrobromide
HTR4: 5-hydroxytryptamine (serotonin) receptor 40.41667Clozapine
0.23774HTR7: 5-hydroxytryptamine (serotonin) receptor 7 (adenylate cyclase-coupled)
206NNNFenoldopam mesylate
DRD3: dopamine receptor D30.36842Haloperidol
0.23823ADRA2A: alpha-2A adrenergic receptor
207NNYSulprostone
PTGER2: prostaglandin E receptor 2 (subtype EP2), 53kDa0.42500Alprostadil
0.17595PTGER1: prostaglandin E receptor 1 (subtype EP1), 42kDa
210NNNSilodosin
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.40909Thiethylperazine
0.18839ADRA1B: alpha-1B adrenergic receptor
217NNNPindolol
DRD5: dopamine receptor D50.34483Chlorpromazine
0.24367HTR4: 5-hydroxytryptamine (serotonin) receptor 4
233NNNPropiomazine
ADRB1: beta-1 adrenergic receptor0.46875Denopamine
0.24984DRD1: dopamine receptor D1
237NNNPindolol
HRH1: histamine receptor H10.37037Diphenhydramine
0.19168HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
253NNNMetoclopramide
ADRB1: beta-1 adrenergic receptor0.41667Amiodarone
0.23627HTR1B: 5-hydroxytryptamine (serotonin) receptor 1B
256NNNBrimonidine tartrate
ADRA1D: alpha-1D adrenergic receptor0.42857Epinephrine bitartrate
0.19423ADRA2C: alpha-2C adrenergic receptor
257YYNAripiprazole
HTR6: 5-hydroxytryptamine (serotonin) receptor 60.47222Clozapine
0.20115HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A
259NNNCaffeine
GPR109A: G protein-coupled receptor 109A0.15000Niacin
0.21659P2RY1: purinergic receptor P2Y, G-protein coupled, 1
268NYYDipivefrin
ADRB2: beta-2 adrenergic receptor0.48918Bitolterol mesylate
0.15399ADRA2A: alpha-2A adrenergic receptor
273NNNMetoclopramide
ADRA1B: alpha-1B adrenergic receptor0.40000Tamsulosin hydrochloride
0.24749HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
278NNNMetoclopramide
ADRB3: beta-3 adrenergic receptor0.39286Bupranolol hydrochloride
0.23779HTR6: 5-hydroxytryptamine (serotonin) receptor 6
279NNNPropiomazine
HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A0.39474Spiperone
0.24883DRD2: dopamine receptor D2
282NNNGuanfacine hydrochloride
ADRA1D: alpha-1D adrenergic receptor0.40909Clonidine hydrochloride
0.19423ADRA2C: alpha-2C adrenergic receptor
285NNNTravoprost
PTGIR: prostaglandin I2 receptor (IP)0.41667Dinoprost tromethamine
0.16339PTGFR: prostaglandin F receptor (FP)
289NNNPropiomazine
HTR6: 5-hydroxytryptamine (serotonin) receptor 60.38235Clozapine
0.24119DRD1: dopamine receptor D1
295NNNNedocromil
LTB4R: leukotriene B4 receptor0.21429Zafirlukast
0.18381CYSLTR1: cysteinyl leukotriene receptor 1
296NNNZafirlukast
PTGDR: prostaglandin D2 receptor (DP)0.21429Nedocromil
0.052938LTB4R: leukotriene B4 receptor
300YNNSumatriptan
DRD4: dopamine receptor D40.37500Propiomazine
0.24653HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
301NNNVerapamil
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.42105Chlorpromazine
0.18839ADRA1B: alpha-1B adrenergic receptor
304NNNMetoclopramide
ADRA2B: alpha-2B adrenergic receptor0.33333Guanfacine hydrochloride
0.24344HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
306NNNPindolol
HRH4: histamine receptor H40.37037Diphenhydramine
0.19094HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
311NNNMetoclopramide
ADRA1D: alpha-1D adrenergic receptor0.40000Tamsulosin hydrochloride
0.22669HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
314NNNLatanoprost
PTGIR: prostaglandin I2 receptor (IP)0.40000Dinoprostone
0.16339PTGFR: prostaglandin F receptor (FP)
320NNNRiluzole
GPRC6A: G protein-coupled receptor, family C, group 6, member A0.083333Lysine hydrochloride
0.18838GRM3: glutamate receptor, metabotropic 3
321NNNPindolol
CHRM2: cholinergic receptor, muscarinic 20.35714Promethazine
0.19911HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
323NNNPropiomazine
ADRB3: beta-3 adrenergic receptor0.43750Dobutamine
0.23650ADRA1B: alpha-1B adrenergic receptor
326NNNCarvedilol
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.42857Promethazine
0.19131ADRB3: beta-3 adrenergic receptor
333NNNSumatriptan
CHRM1: cholinergic receptor, muscarinic 10.37931Promethazine
0.21367HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
345NNNMetoclopramide
DRD5: dopamine receptor D50.32258Chlorpromazine
0.24367HTR4: 5-hydroxytryptamine (serotonin) receptor 4
349NNNCarboprost tromethamine
PTGER3: prostaglandin E receptor 3 (subtype EP3)0.35623Misoprostol
0.20058PTGER1: prostaglandin E receptor 1 (subtype EP1), 42kDa
358NNNCaffeine
MTNR1A: melatonin receptor 1A0.28000Agomelatine
0.15074ADORA2B: adenosine A2b receptor
359NNNSilodosin
ADRA2B: alpha-2B adrenergic receptor0.38636Haloperidol
0.19075ADRA1A: alpha-1A adrenergic receptor
360NNNEletriptan hydrobromide
HRH1: histamine receptor H10.47222Prochlorperazine
0.19168HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
375NNNNedocromil
LTB4R2: leukotriene B4 receptor 20.21429Zafirlukast
0.11219CYSLTR1: cysteinyl leukotriene receptor 1
379NNNEletriptan hydrobromide
CHRM1: cholinergic receptor, muscarinic 10.48571Methixene hydrochloride
0.21367HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
380NNNVerapamil
ADRB1: beta-1 adrenergic receptor0.47368Denopamine
0.23215ADRA1A: alpha-1A adrenergic receptor
382NNNRiluzole
GABBR1: gamma-aminobutyric acid (GABA) B receptor, 10.26087Baclofen
0.056171GRM4: glutamate receptor, metabotropic 4
383NNNCaffeine
LTB4R: leukotriene B4 receptor0.17021Zafirlukast
0.16987P2RY1: purinergic receptor P2Y, G-protein coupled, 1
385NNNCaffeine
OPRD1: opioid receptor, delta 10.23333Oxycodone
0.20964P2RY4: pyrimidinergic receptor P2Y, G-protein coupled, 4
387NNNSumatriptan
ADRA1B: alpha-1B adrenergic receptor0.44118Tamsulosin hydrochloride
0.24749HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
392NYNAripiprazole
ADRA2B: alpha-2B adrenergic receptor0.47222Clozapine
0.24344HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
396NYNCyproheptadine hydrochloride
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.35849Clozapine
0.18839ADRA1B: alpha-1B adrenergic receptor
397NNNPrazosin hydrochloride
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.41667Olanzapine
0.18839ADRA1B: alpha-1B adrenergic receptor
400NNNEpinastine hydrochloride
CHRM1: cholinergic receptor, muscarinic 10.48276Clozapine
0.20344HRH1: histamine receptor H1
407NNNEglumegad
GPRC6A: G protein-coupled receptor, family C, group 6, member A0.33333Lysine acetate
0.18838GRM3: glutamate receptor, metabotropic 3
408NNNSumatriptan
ADRB1: beta-1 adrenergic receptor0.41935Bretylium tosylate
0.23627HTR1B: 5-hydroxytryptamine (serotonin) receptor 1B
417NNNFamotidine
HRH1: histamine receptor H10.14706Diphenhydramine
0.17437HRH3: histamine receptor H3
418NNNAstemizole
ADRA1A: alpha-1A adrenergic receptor0.48780Perphenazine
0.16141HRH4: histamine receptor H4
420NNNCaffeine
SSTR1: somatostatin receptor 10.089744Octreotide
0.22075CXCR1: chemokine (C-X-C motif) receptor 1
423YNNNifedipine
CHRM1: cholinergic receptor, muscarinic 10.30556Homatropine methylbromide
0.19188ADRA2A: alpha-2A adrenergic receptor
427NNNNifedipine
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.25641Propiomazine
0.19131ADRB3: beta-3 adrenergic receptor
429NNNCaffeine
EDNRA: endothelin receptor type A0.17391Bosentan
0.13544CXCR1: chemokine (C-X-C motif) receptor 1
431NNNFenoldopam mesylate
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.39394Mirtazapine
0.18605DRD1: dopamine receptor D1
433NNNMetoclopramide
HRH4: histamine receptor H40.25806Diphenhydramine
0.19094HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
434NNNCarvedilol
CXCR1: chemokine (C-X-C motif) receptor 10.44444Trimipramine
0.12052ADRA1A: alpha-1A adrenergic receptor
438NNNAripiprazole
HTR4: 5-hydroxytryptamine (serotonin) receptor 40.47222Clozapine
0.20265HTR2C: 5-hydroxytryptamine (serotonin) receptor 2C
439NNNCaffeine
GPR109B: G protein-coupled receptor 109B0.21429Metoclopramide
0.21186P2RY1: purinergic receptor P2Y, G-protein coupled, 1
440NNNSumatriptan
HRH4: histamine receptor H40.37931Promethazine
0.19094HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
447NNNEletriptan hydrobromide
ADRA1B: alpha-1B adrenergic receptor0.44118Mianserin hydrochloride
0.24749HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
448NNNCaffeine
EDNRB: endothelin receptor type B0.17391Bosentan
0.13847P2RY1: purinergic receptor P2Y, G-protein coupled, 1
451NNNPromethazine
ADRB1: beta-1 adrenergic receptor0.46667Bretylium tosylate
0.23215ADRA1A: alpha-1A adrenergic receptor
452NNNSumatriptan
ADRA1D: alpha-1D adrenergic receptor0.44118Tamsulosin hydrochloride
0.22669HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
454NNNAgomelatine
HTR4: 5-hydroxytryptamine (serotonin) receptor 40.48148Tegaserod
0.20265HTR2C: 5-hydroxytryptamine (serotonin) receptor 2C
456NNNCaffeine
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.25926Sumatriptan
0.13508ADORA2B: adenosine A2b receptor
457NNNSilodosin
ADRA2A: alpha-2A adrenergic receptor0.38636Haloperidol
0.19136ADRA1B: alpha-1B adrenergic receptor
459NNNCaffeine
CNR1: cannabinoid receptor 1 (brain)0.23333Dronabinol
0.12689ADORA2B: adenosine A2b receptor
460NNNSumatriptan
ADRA2B: alpha-2B adrenergic receptor0.41379Chlorpromazine
0.24344HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
466NNNSolifenacin succinate
HRH1: histamine receptor H10.48718Mequitazine
0.20344CHRM1: cholinergic receptor, muscarinic 1
469NNNMethoxamine hydrochloride
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.38461Metoclopramide
0.18839ADRA1B: alpha-1B adrenergic receptor
470NNNMetoclopramide
HRH1: histamine receptor H10.33333Propiomazine
0.20344CHRM1: cholinergic receptor, muscarinic 1
473NNNSumatriptan
GPR109B: G protein-coupled receptor 109B0.33333Metoclopramide
0.070289HTR4: 5-hydroxytryptamine (serotonin) receptor 4
476NNNSumatriptan
ADRB3: beta-3 adrenergic receptor0.40741Pindolol
0.23779HTR6: 5-hydroxytryptamine (serotonin) receptor 6
477NNNEletriptan hydrobromide
ADRA1D: alpha-1D adrenergic receptor0.44118Mianserin hydrochloride
0.22669HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
480NNNCaffeine
SSTR30.094118Octreotide acetate
0.19590CXCR1: chemokine (C-X-C motif) receptor 1
481NNNCaffeine
SSTR5: somatostatin receptor 50.094118Octreotide acetate
0.21230CXCR1: chemokine (C-X-C motif) receptor 1
487NNNCarvedilol
HRH1: histamine receptor H10.42857Promethazine
0.17178ADRA2A: alpha-2A adrenergic receptor
493NNNPropiomazine
HTR7: 5-hydroxytryptamine (serotonin) receptor 7 (adenylate cyclase-coupled)0.39474Spiperone
0.24985ADRA1A: alpha-1A adrenergic receptor
494NYNChlorpromazine phenolphthalinate
DRD1: dopamine receptor D10.46667Chlorpromazine
0.17607ADRA2A: alpha-2A adrenergic receptor
507NNNNilutamide
CXCR1: chemokine (C-X-C motif) receptor 10.34483Aminoglutethimide
0.12052ADRA1A: alpha-1A adrenergic receptor
510NNNPalmitic acid
PTGIR: prostaglandin I2 receptor (IP)0.48276Alprostadil
0.069739RHO: rhodopsin
512NNNEletriptan hydrobromide
ADRA2B: alpha-2B adrenergic receptor0.42857Olanzapine
0.24344HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
513NNNCaffeine
RHO: rhodopsin0.032258Palmitic acid
0.13510ADORA2B: adenosine A2b receptor
525NNNCyproheptadine hydrochloride
ADRA2B: alpha-2B adrenergic receptor0.37500Chlorpromazine hibenzate
0.19075ADRA1A: alpha-1A adrenergic receptor
526NNNVerapamil
HRH1: histamine receptor H10.39024Propiomazine
0.21072CHRM2: cholinergic receptor, muscarinic 2
533NNNOlanzapine
ADORA2B: adenosine A2b receptor0.25000Theophylline
0.19234ADRB2: beta-2 adrenergic receptor
534NNNPindolol
CHRM4: cholinergic receptor, muscarinic 40.35714Promethazine
0.19755HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
537NNNEpinastine hydrochloride
ADRB3: beta-3 adrenergic receptor0.35484Olanzapine
0.24769HRH2: histamine receptor H2
538NNNDenopamine
ADRA1A: alpha-1A adrenergic receptor0.47368Verapamil
0.23215ADRB1: beta-1 adrenergic receptor
539NNNSumatriptan
DRD5: dopamine receptor D50.41379Chlorpromazine
0.24367HTR4: 5-hydroxytryptamine (serotonin) receptor 4
542NNNCaffeine
GPRC5A: G protein-coupled receptor, family C, group 5, member A0.090909Tretinoin
0.040625ADORA3: adenosine A3 receptor
544NNNCaffeine
NTSR2: neurotensin receptor 20.12195Levocabastine hydrochloride
0.098693ADORA2B: adenosine A2b receptor
545NNNPalmitic acid
GPRC6A: G protein-coupled receptor, family C, group 6, member A0.33333Lysine acetate
0.015237RHO: rhodopsin
548NNNAmlexanox
PTGDR: prostaglandin D2 receptor (DP)0.44118Nedocromil
0.032702CYSLTR1: cysteinyl leukotriene receptor 1
549NNNRizatriptan benzoate
HRH1: histamine receptor H10.46154Doxylamine succinate
0.18251HTR1B: 5-hydroxytryptamine (serotonin) receptor 1B
551NNNIloprost
PTGER3: prostaglandin E receptor 3 (subtype EP3)0.35897Misoprostol
0.20058PTGER1: prostaglandin E receptor 1 (subtype EP1), 42kDa
552YNNRisperidone
HTR7: 5-hydroxytryptamine (serotonin) receptor 7 (adenylate cyclase-coupled)0.39474Clozapine
0.24985ADRA1A: alpha-1A adrenergic receptor
553NNNPromethazine
ADRB2: beta-2 adrenergic receptor0.46667Bretylium tosylate
0.24577ADRA1A: alpha-1A adrenergic receptor
560NNNMethoxamine hydrochloride
ADRB1: beta-1 adrenergic receptor0.45833Atenolol
0.23215ADRA1A: alpha-1A adrenergic receptor
565NNNVerapamil
ADRB2: beta-2 adrenergic receptor0.39655Metoprolol tartrate
0.24577ADRA1A: alpha-1A adrenergic receptor
566NNNAlprazolam
HRH1: histamine receptor H10.45161Clozapine
0.053108CXCR1: chemokine (C-X-C motif) receptor 1
567NNNBretylium tosylate
HRH1: histamine receptor H10.46875Triprolidine hydrochloride
0.13611ADRB2: beta-2 adrenergic receptor
572NNNBosentan
GPR37L1: G protein-coupled receptor 37 like 10.38983Imatinib mesilate
0.14980EDNRA: endothelin receptor type A
574NNNChlorpromazine hibenzate
ADRA1D: alpha-1D adrenergic receptor0.40000Propiomazine
0.19423ADRA2C: alpha-2C adrenergic receptor
576NYNAripiprazole
ADRA1B: alpha-1B adrenergic receptor0.49391Spiperone
0.23485HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
578NNNPrazosin hydrochloride
HRH1: histamine receptor H10.41667Olanzapine
0.17178ADRA2A: alpha-2A adrenergic receptor
581NNNCaffeine
LTB4R2: leukotriene B4 receptor 20.17021Zafirlukast
0.12916P2RY6: pyrimidinergic receptor P2Y, G-protein coupled, 6
582NNNCaffeine
PTGDR: prostaglandin D2 receptor (DP)0.28125Nedocromil
0.072107ADORA2B: adenosine A2b receptor
586NNNAripiprazole
ADRA1D: alpha-1D adrenergic receptor0.49391Spiperone
0.22542HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
592NNNOlanzapine
ADORA1: adenosine A1 receptor0.24138Caffeine
0.16314DRD1: dopamine receptor D1
597NNNPromethazine
ADRB3: beta-3 adrenergic receptor0.42857Carvedilol
0.23647ADRA1A: alpha-1A adrenergic receptor
598NNNCaffeine
GPR37L1: G protein-coupled receptor 37 like 10.16667Imatinib mesilate
0.068153LPAR6: lysophosphatidic acid receptor 6
599NNNAmlexanox
HRH1: histamine receptor H10.44118Nedocromil
0.058535CYSLTR1: cysteinyl leukotriene receptor 1
601NNNPrazosin hydrochloride
CHRM1: cholinergic receptor, muscarinic 10.42500Pirenzepine hydrochloride
0.19188ADRA2A: alpha-2A adrenergic receptor
603NNNDimenhydrinate
ADORA2A: adenosine A2a receptor0.43182Aminophylline
0.10258HRH1: histamine receptor H1
604YYNCisapride
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.46154Prochlorperazine
0.18539HTR4: 5-hydroxytryptamine (serotonin) receptor 4
605NNNApafant
DRD2: dopamine receptor D20.40000Prochlorperazine
0.062824PTAFR: platelet-activating factor receptor
607NNNAgomelatine
DRD2: dopamine receptor D20.46154Metoclopramide
0.20058HTR2C: 5-hydroxytryptamine (serotonin) receptor 2C
609NNNPalmitic acid
PTGER2: prostaglandin E receptor 2 (subtype EP2), 53kDa0.48276Alprostadil
0.049640RHO: rhodopsin
611NNNClozapine
MTNR1A: melatonin receptor 1A0.28125Agomelatine
0.14358HTR4: 5-hydroxytryptamine (serotonin) receptor 4
612NNNAmiodarone
DRD2: dopamine receptor D20.44737Propiomazine
0.18564ADRA1A: alpha-1A adrenergic receptor
614NNNMethoxamine hydrochloride
ADRA2A: alpha-2A adrenergic receptor0.42857Epinephrine hydrochloride
0.19136ADRA1B: alpha-1B adrenergic receptor
615NNNIrbesartan
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.48780Spiperone
0.10570AGTR1: angiotensin II receptor, type 1
620YNNZafirlukast
PTAFR: platelet-activating factor receptor0.26316Apafant
0.24638CYSLTR1: cysteinyl leukotriene receptor 1
625NNNEletriptan hydrobromide
CHRM2: cholinergic receptor, muscarinic 20.48571Methixene hydrochloride
0.19911HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
626NNNNilutamide
ADRB1: beta-1 adrenergic receptor0.31034Isoproterenol hydrochloride
0.23215ADRA1A: alpha-1A adrenergic receptor
627NYNTegaserod
HTR2C: 5-hydroxytryptamine (serotonin) receptor 2C0.48148Agomelatine
0.20265HTR4: 5-hydroxytryptamine (serotonin) receptor 4
629NNNPentobarbital
CXCR1: chemokine (C-X-C motif) receptor 10.37500Hexobarbital
0.15780GPR109B: G protein-coupled receptor 109B
633NNNEletriptan hydrobromide
DRD4: dopamine receptor D40.44737Thiethylperazine
0.24653HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
636NNNChlorpromazine phenolphthalinate
ADRA1D: alpha-1D adrenergic receptor0.34286Cyproheptadine hydrochloride
0.19423ADRA2C: alpha-2C adrenergic receptor
637NNYDipivefrin
ADRB1: beta-1 adrenergic receptor0.42424Metipranolol
0.20800ADRA2A: alpha-2A adrenergic receptor
638NNNCaffeine
CCKAR: cholecystokinin A receptor0.069307Ceruletide
0.13320ADORA2B: adenosine A2b receptor
639NNNPindolol
CHRM3: cholinergic receptor, muscarinic 30.35714Promethazine
0.15935HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
648YYNRisperidone
HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A0.39474Clozapine
0.24550ADRA1A: alpha-1A adrenergic receptor
649NNNPropiomazine
ADRA2C: alpha-2C adrenergic receptor0.40000Chlorpromazine hibenzate
0.24052DRD4: dopamine receptor D4
657NNNCocaine
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.31250Mirtazapine
0.18620DRD3: dopamine receptor D3
660NNNHomatropine methylbromide
DRD4: dopamine receptor D40.29412Olanzapine
0.17454CHRM1: cholinergic receptor, muscarinic 1
662NNNAgomelatine
HTR6: 5-hydroxytryptamine (serotonin) receptor 60.46154Sumatriptan
0.19328HTR2C: 5-hydroxytryptamine (serotonin) receptor 2C
663NNNChlorpromazine phenolphthalinate
DRD5: dopamine receptor D50.46667Chlorpromazine
0.15748ADRA2A: alpha-2A adrenergic receptor
665NNNCaffeine
AVPR1A: arginine vasopressin receptor 1A0.12766Conivaptan hydrochloride
0.11011CXCR1: chemokine (C-X-C motif) receptor 1
666NNNEpinastine hydrochloride
DRD3: dopamine receptor D30.48276Loxapine
0.23823ADRA2A: alpha-2A adrenergic receptor
667NNNCaffeine
OPRK1: opioid receptor, kappa 10.23333Oxycodone
0.21114LPAR6: lysophosphatidic acid receptor 6
669NNNEletriptan hydrobromide
CHRM3: cholinergic receptor, muscarinic 30.48571Methixene hydrochloride
0.15935HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
670NNNEpinephrine bitartrate
HRH1: histamine receptor H10.38889Chlorpheniramine maleate
0.17178ADRA2A: alpha-2A adrenergic receptor
673YNNClozapine
ADORA3: adenosine A3 receptor0.15625Caffeine
0.16830HTR4: 5-hydroxytryptamine (serotonin) receptor 4
675NNNOxycodone
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.32500Risperidone
0.11643OPRK1: opioid receptor, kappa 1
678NNNEpinephrine hydrochloride
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.39130Pindolol
0.19131ADRB3: beta-3 adrenergic receptor
682NNNCaffeine
AVPR2: arginine vasopressin receptor 20.12766Conivaptan hydrochloride
0.10409P2RY12: purinergic receptor P2Y, G-protein coupled, 12
684NNNCaffeine
GABBR1: gamma-aminobutyric acid (GABA) B receptor, 10.076923Baclofen
0.024835P2RY12: purinergic receptor P2Y, G-protein coupled, 12
688NNNCaffeine
ADRA1A: alpha-1A adrenergic receptor0.25926Promethazine
0.14755ADORA2B: adenosine A2b receptor
691NNNDimenhydrinate
ADORA1: adenosine A1 receptor0.43182Aminophylline
0.10999HRH1: histamine receptor H1
693NNNAmiodarone
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.44737Propiomazine
0.19040ADRB1: beta-1 adrenergic receptor
695NNNEpinastine hydrochloride
HRH4: histamine receptor H40.48276Clozapine
0.16558ADRA1B: alpha-1B adrenergic receptor
697NNNOlanzapine
ADORA2A: adenosine A2a receptor0.24138Caffeine
0.18127ADRB3: beta-3 adrenergic receptor
698NNNClozapine
ADORA2B: adenosine A2b receptor0.16129Theophylline
0.17980HTR7: 5-hydroxytryptamine (serotonin) receptor 7 (adenylate cyclase-coupled)
699NNNDexmedetomidine
HRH1: histamine receptor H10.41667Diphenhydramine
0.17178ADRA2A: alpha-2A adrenergic receptor
700NNNOlanzapine
OPRM1: opioid receptor, mu 10.44118Sufentanil
0.15246ADRB2: beta-2 adrenergic receptor
701NNNCaffeine
CCKBR: cholecystokinin B receptor0.069307Ceruletide
0.10948CXCR1: chemokine (C-X-C motif) receptor 1
703NNNCeruletide
TRHR: thyrotropin-releasing hormone receptor0.24762Protirelin tartrate hydrate
0.15446CCKAR: cholecystokinin A receptor
704NNNCaffeine
SSTR20.094118Octreotide acetate
0.21327LPAR6: lysophosphatidic acid receptor 6
705YNNNifedipine
CHRM2: cholinergic receptor, muscarinic 20.30556Homatropine methylbromide
0.16943ADRA2A: alpha-2A adrenergic receptor
709NNNClozapine
ADORA1: adenosine A1 receptor0.15625Caffeine
0.17450HTR4: 5-hydroxytryptamine (serotonin) receptor 4
711NNNPindolol
ADORA2B: adenosine A2b receptor0.28000Enprofylline
0.19234ADRB2: beta-2 adrenergic receptor
713NNNPindolol
CHRM5: cholinergic receptor, muscarinic 50.35714Promethazine
0.16744HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
714NNNCarvedilol
HTR2C: 5-hydroxytryptamine (serotonin) receptor 2C0.41176Pindolol
0.19362ADRA1A: alpha-1A adrenergic receptor
716NNNMetoclopramide
MTNR1A: melatonin receptor 1A0.46154Agomelatine
0.14358HTR4: 5-hydroxytryptamine (serotonin) receptor 4
717NNNBrimonidine tartrate
ADRA1B: alpha-1B adrenergic receptor0.42857Epinephrine bitartrate
0.19685ADRA2C: alpha-2C adrenergic receptor
718NNNRiluzole
GPRC5A: G protein-coupled receptor, family C, group 5, member A0Tretinoin
0.048612GRM2: glutamate receptor, metabotropic 2
719NNNEpinastine hydrochloride
CHRM2: cholinergic receptor, muscarinic 20.48276Clozapine
0.21072HRH1: histamine receptor H1
721NNNPindolol
HRH3: histamine receptor H30.37037Diphenhydramine
0.21026ADRA2A: alpha-2A adrenergic receptor
722NNNPrazosin hydrochloride
CHRM2: cholinergic receptor, muscarinic 20.41861Cisapride
0.16943ADRA2A: alpha-2A adrenergic receptor
723NNNOxymetazoline hydrochloride
ADRB3: beta-3 adrenergic receptor0.39286Bupranolol hydrochloride
0.23650ADRA1B: alpha-1B adrenergic receptor
724NNNAncriviroc
DRD2: dopamine receptor D20.40909Haloperidol
0.067092CCR5: chemokine (C-C motif) receptor 5
725NNNClopidogrel bisulfate
ADRA2A: alpha-2A adrenergic receptor0.40541Fenoldopam mesylate
0.050826P2RY12: purinergic receptor P2Y, G-protein coupled, 12
726NYNCabergoline
DRD1: dopamine receptor D10.32558Propiomazine
0.17500DRD2: dopamine receptor D2
728NNNCyproheptadine hydrochloride
ADRA2A: alpha-2A adrenergic receptor0.37500Chlorpromazine hibenzate
0.19136ADRA1B: alpha-1B adrenergic receptor
729NNNClopidogrel bisulfate
HRH1: histamine receptor H10.39394Cyclizine
0.053949P2RY12: purinergic receptor P2Y, G-protein coupled, 12
730NNNPrazosin hydrochloride
ADRB3: beta-3 adrenergic receptor0.41667Olanzapine
0.23650ADRA1B: alpha-1B adrenergic receptor
731NNNAmlexanox
LTB4R: leukotriene B4 receptor0.26000Zafirlukast
0.18381CYSLTR1: cysteinyl leukotriene receptor 1
732NNNEletriptan hydrobromide
HRH4: histamine receptor H40.44186Astemizole
0.19094HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
734NNNDexmedetomidine
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.40000Promethazine
0.13659ADRA2A: alpha-2A adrenergic receptor
735NNNPramipexole hydrochloride
HRH2: histamine receptor H20.26667Nizatidine
0.17831DRD3: dopamine receptor D3
736NYNEpinastine hydrochloride
HTR7: 5-hydroxytryptamine (serotonin) receptor 7 (adenylate cyclase-coupled)0.48276Clozapine
0.24985ADRA1A: alpha-1A adrenergic receptor
738NYNPramipexole hydrochloride
DRD1: dopamine receptor D10.23529Prochlorperazine
0.20484DRD3: dopamine receptor D3
739NNNMesoridazine
OPRD1: opioid receptor, delta 10.37949Pimozide
0.12709DRD1: dopamine receptor D1
740NNNZafirlukast
CCR5: chemokine (C-C motif) receptor 50.30508Ancriviroc
0.21623CYSLTR2: cysteinyl leukotriene receptor 2
741NNNPrazosin hydrochloride
DRD3: dopamine receptor D30.41667Olanzapine
0.23823ADRA2A: alpha-2A adrenergic receptor
743NNNCaffeine
HRH1: histamine receptor H10.34286Dimenhydrinate
0.10999ADORA1: adenosine A1 receptor
744NNNEpinephrine hydrochloride
CXCR1: chemokine (C-X-C motif) receptor 10.28571Trimipramine
0.12052ADRA1A: alpha-1A adrenergic receptor
745NNNImatinib mesilate
DRD2: dopamine receptor D20.40816Thiethylperazine
0.065803GPR37L1: G protein-coupled receptor 37 like 1
747NNNClozapine
CCKAR: cholecystokinin A receptor0.13592Ceruletide
0.13795HTR4: 5-hydroxytryptamine (serotonin) receptor 4
748NNNBaclofen
GPRC6A: G protein-coupled receptor, family C, group 6, member A0.31579Lysine hydrochloride
0.029235GABBR1: gamma-aminobutyric acid (GABA) B receptor, 1
752NNNCyproheptadine hydrochloride
ADRA2C: alpha-2C adrenergic receptor0.37500Chlorpromazine hibenzate
0.19685ADRA1B: alpha-1B adrenergic receptor
758NNNClonidine
ADRB3: beta-3 adrenergic receptor0.24138Olanzapine
0.23650ADRA1B: alpha-1B adrenergic receptor
759NNNClopidogrel bisulfate
CXCR1: chemokine (C-X-C motif) receptor 10.37143Trimipramine
0.15447P2RY12: purinergic receptor P2Y, G-protein coupled, 12
760NNNLatanoprost
ADRB2: beta-2 adrenergic receptor0.42105Betaxolol hydrochloride
0.040226PTGFR: prostaglandin F receptor (FP)
762NNNMethoxamine hydrochloride
ADRA2B: alpha-2B adrenergic receptor0.42857Epinephrine hydrochloride
0.19075ADRA1A: alpha-1A adrenergic receptor
763NNNCaffeine
TBXA2R: thromboxane A2 receptor0.12121Daltroban
0.086403P2RY6: pyrimidinergic receptor P2Y, G-protein coupled, 6
765NNNBethanidine sulfate
ADRB2: beta-2 adrenergic receptor0.46154Bretylium tosylate
0.24577ADRA1A: alpha-1A adrenergic receptor
766NNNDezocine
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.37500Mesoridazine
0.11643OPRK1: opioid receptor, kappa 1
772NNNTamsulosin hydrochloride
ADRA2B: alpha-2B adrenergic receptor0.47059Chlorpromazine
0.19075ADRA1A: alpha-1A adrenergic receptor
776NNNBethanidine sulfate
HRH2: histamine receptor H20.28571Ranitidine
0.23944ADRA1A: alpha-1A adrenergic receptor
778NNNTegaserod
HTR5A: 5-hydroxytryptamine (serotonin) receptor 5A0.44828Sumatriptan
0.20005HTR4: 5-hydroxytryptamine (serotonin) receptor 4
779NNNAtropine
DRD4: dopamine receptor D40.26471Olanzapine
0.17454CHRM1: cholinergic receptor, muscarinic 1
783NNNPindolol
MTNR1A: melatonin receptor 1A0.44000Agomelatine
0.14358HTR4: 5-hydroxytryptamine (serotonin) receptor 4
784NNNOxymetazoline hydrochloride
ADRB1: beta-1 adrenergic receptor0.39286Bupranolol hydrochloride
0.23215ADRA1A: alpha-1A adrenergic receptor
785NNNSilodosin
ADRB1: beta-1 adrenergic receptor0.43478Amiodarone
0.23215ADRA1A: alpha-1A adrenergic receptor
790NNNPhentolamine mesylate
ADRB2: beta-2 adrenergic receptor0.42857Bretylium tosylate
0.24577ADRA1A: alpha-1A adrenergic receptor
791NNNNorgestrel
OPRM1: opioid receptor, mu 10.33333Naltrexone
0.14177ADRA1A: alpha-1A adrenergic receptor
793NNNPromethazine
HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A0.38710Clozapine
0.24883DRD2: dopamine receptor D2
799NNNSumatriptan
CHRM2: cholinergic receptor, muscarinic 20.37931Promethazine
0.19911HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
801NNNClozapine
TRHR: thyrotropin-releasing hormone receptor0.21429Montirelin
0.13255ADRA1A: alpha-1A adrenergic receptor
804NNNSumatriptan
HRH1: histamine receptor H10.37931Promethazine
0.19168HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F
805NNNNicotine
CXCR1: chemokine (C-X-C motif) receptor 10.31818Metyrapone
0.15780GPR109B: G protein-coupled receptor 109B
806NNNHomatropine methylbromide
HRH1: histamine receptor H10.36111Loratadine
0.21072CHRM2: cholinergic receptor, muscarinic 2
807NNNFenoldopam mesylate
ADRB1: beta-1 adrenergic receptor0.44118Dobutamine hydrochloride
0.24984DRD1: dopamine receptor D1
809NNNClozapine
CCKBR: cholecystokinin B receptor0.13592Ceruletide
0.12538HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A
812NNNTegaserod
HTR6: 5-hydroxytryptamine (serotonin) receptor 60.44828Sumatriptan
0.21711HTR4: 5-hydroxytryptamine (serotonin) receptor 4
814NNNAncriviroc
HRH1: histamine receptor H10.40000Loratadine
0.076313CCR5: chemokine (C-C motif) receptor 5
815NYNLisuride maleate
DRD1: dopamine receptor D10.28261Mesoridazine
0.17500DRD2: dopamine receptor D2
818NNNNicotine
CHRM1: cholinergic receptor, muscarinic 10.39130Cyclizine
0.054306GPR109B: G protein-coupled receptor 109B
823NNNAmlexanox
AGTR1: angiotensin II receptor, type 10.38461Valsartan
0.21175CYSLTR1: cysteinyl leukotriene receptor 1
824NNNAmlexanox
LTB4R2: leukotriene B4 receptor 20.26000Zafirlukast
0.11219CYSLTR1: cysteinyl leukotriene receptor 1
826NNNRiluzole
PTGDR: prostaglandin D2 receptor (DP)0.16667Nedocromil
0.017518GRM2: glutamate receptor, metabotropic 2
827NNYChlorpromazine phenolphthalinate
HRH1: histamine receptor H10.39286Dimenhydrinate
0.17178ADRA2A: alpha-2A adrenergic receptor
828NNNBretylium tosylate
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.46667Promethazine
0.19040ADRB1: beta-1 adrenergic receptor
832NNNClozapine
ADORA2A: adenosine A2a receptor0.15625Caffeine
0.18108HTR4: 5-hydroxytryptamine (serotonin) receptor 4
833NYNBromocriptine mesylate
DRD1: dopamine receptor D10.27586Fenoldopam mesylate
0.17500DRD2: dopamine receptor D2
835NNNRenzapride
HTR6: 5-hydroxytryptamine (serotonin) receptor 60.44828Metoclopramide
0.21711HTR4: 5-hydroxytryptamine (serotonin) receptor 4
836NNNTropicamide
HRH1: histamine receptor H10.48148Diphenhydramine
0.21072CHRM2: cholinergic receptor, muscarinic 2
838NNNDezocine
DRD1: dopamine receptor D10.37500Mesoridazine
0.13442OPRK1: opioid receptor, kappa 1
839NNNPindolol
ADORA2A: adenosine A2a receptor0.23333Ambuphylline
0.18127ADRB3: beta-3 adrenergic receptor
840NNNBrimonidine tartrate
ADRA1A: alpha-1A adrenergic receptor0.42857Epinephrine bitartrate
0.19610ADRA2C: alpha-2C adrenergic receptor
841NNNEpinastine hydrochloride
ADRB1: beta-1 adrenergic receptor0.35484Olanzapine
0.23662HRH2: histamine receptor H2
843NNNLevocabastine hydrochloride
CHRM1: cholinergic receptor, muscarinic 10.45903Trospium chloride
0.20344HRH1: histamine receptor H1
844NNNClozapine
OPRD1: opioid receptor, delta 10.42500Pimozide
0.14993HTR4: 5-hydroxytryptamine (serotonin) receptor 4
845NNNPhentolamine mesylate
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.40541Mesoridazine
0.18839ADRA1B: alpha-1B adrenergic receptor
850NNNSpironolactone
OPRM1: opioid receptor, mu 10.26829Oxycodone
0.22103AGTR1: angiotensin II receptor, type 1
851NNNRiluzole
ADRA1A: alpha-1A adrenergic receptor0.40909Methoxamine hydrochloride
0.016893GRM1: glutamate receptor, metabotropic 1
852NNNCisapride
HRH1: histamine receptor H10.46667Astemizole
0.21072CHRM2: cholinergic receptor, muscarinic 2
853NNNOlanzapine
ADORA3: adenosine A3 receptor0.24138Caffeine
0.14751ADRA1B: alpha-1B adrenergic receptor
854NNNClozapine
CNR1: cannabinoid receptor 1 (brain)0.21053Dronabinol
0.12220ADRA1A: alpha-1A adrenergic receptor
859NNNCocaine
CXCR1: chemokine (C-X-C motif) receptor 10.38235Nifedipine
0.19826OPRK1: opioid receptor, kappa 1
860YNNSpiperone
DRD4: dopamine receptor D40.47368Thiethylperazine
0.24653HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A
861NNNPropiomazine
HTR5A: 5-hydroxytryptamine (serotonin) receptor 5A0.38235Clozapine
0.24618ADRA1A: alpha-1A adrenergic receptor
863YNNZafirlukast
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.42553Mesoridazine
0.078533CYSLTR1: cysteinyl leukotriene receptor 1
865NNNCaffeine
ADRA2B: alpha-2B adrenergic receptor0.25926Oxymetazoline hydrochloride
0.12114ADORA1: adenosine A1 receptor
866NNNRenzapride
HTR5A: 5-hydroxytryptamine (serotonin) receptor 5A0.44828Metoclopramide
0.20005HTR4: 5-hydroxytryptamine (serotonin) receptor 4
869NNNNifedipine
DRD3: dopamine receptor D30.38235Cocaine
0.23823ADRA2A: alpha-2A adrenergic receptor
871NNYDipivefrin
ADRB3: beta-3 adrenergic receptor0.42424Metipranolol
0.18550ADRA2A: alpha-2A adrenergic receptor
872YNNZafirlukast
HRH1: histamine receptor H10.41509Astemizole
0.082851LTB4R: leukotriene B4 receptor
874NNNGuanabenz
HRH2: histamine receptor H20.25926Epinastine hydrochloride
0.16382ADRA2A: alpha-2A adrenergic receptor
878NNNAgomelatine
ADRA2A: alpha-2A adrenergic receptor0.44444Chlorpromazine
0.15657HTR2C: 5-hydroxytryptamine (serotonin) receptor 2C
883NNNOxymetazoline hydrochloride
CHRM1: cholinergic receptor, muscarinic 10.33333Tolterodine
0.19188ADRA2A: alpha-2A adrenergic receptor
884NNNNedocromil
PTAFR: platelet-activating factor receptor0.20833Apafant
0.24638CYSLTR1: cysteinyl leukotriene receptor 1
885NNNBosentan
AGTR1: angiotensin II receptor, type 10.40385Olmesartan
0.12880EDNRB: endothelin receptor type B
886NNNPhentolamine mesylate
ADRB1: beta-1 adrenergic receptor0.42857Bretylium tosylate
0.23215ADRA1A: alpha-1A adrenergic receptor
887NNNTamsulosin hydrochloride
ADRA2A: alpha-2A adrenergic receptor0.47059Chlorpromazine
0.19136ADRA1B: alpha-1B adrenergic receptor
889NYNChlorpromazine hibenzate
ADRA1A: alpha-1A adrenergic receptor0.40425Perphenazine
0.19610ADRA2C: alpha-2C adrenergic receptor
890NNNTegaserod
HTR1F: 5-hydroxytryptamine (serotonin) receptor 1F0.44828Sumatriptan
0.22464HTR4: 5-hydroxytryptamine (serotonin) receptor 4
893NNNLatanoprost
ADRB1: beta-1 adrenergic receptor0.42105Betaxolol hydrochloride
0.046860PTGFR: prostaglandin F receptor (FP)
895NNNCeruletide
SSTR20.34109Octreotide acetate
0.16860CCKAR: cholecystokinin A receptor
897NNNAmiodarone
HRH1: histamine receptor H10.44737Propiomazine
0.12344ADRA1A: alpha-1A adrenergic receptor
899NNNMetyrapone
CHRM1: cholinergic receptor, muscarinic 10.46154Tropicamide
0.059358CXCR1: chemokine (C-X-C motif) receptor 1
902NNNCarvedilol
CHRM1: cholinergic receptor, muscarinic 10.43243Profenamine hydrochloride
0.19188ADRA2A: alpha-2A adrenergic receptor
904NNNDaltroban
GABBR1: gamma-aminobutyric acid (GABA) B receptor, 10.48000Baclofen
0.012988TBXA2R: thromboxane A2 receptor
906YNNAtropine
HRH1: histamine receptor H10.36667Cyclizine
0.21072CHRM2: cholinergic receptor, muscarinic 2
907NNNEpinastine hydrochloride
HRH3: histamine receptor H30.46429Maprotiline
0.21026ADRA2A: alpha-2A adrenergic receptor
908NNNClozapine
OPRM1: opioid receptor, mu 10.38889Sufentanil
0.15722HTR4: 5-hydroxytryptamine (serotonin) receptor 4
909NNNAncriviroc
OPRM1: opioid receptor, mu 10.40000Sufentanil
0.20189CCR5: chemokine (C-C motif) receptor 5
910NNNAlniditan dihydrochloride
DRD2: dopamine receptor D20.38235Loxapine
0.23462HTR1D: 5-hydroxytryptamine (serotonin) receptor 1D
911NNNEpinephrine bitartrate
CHRM1: cholinergic receptor, muscarinic 10.30769Doxylamine succinate
0.19188ADRA2A: alpha-2A adrenergic receptor
912NNNVerapamil
HTR2C: 5-hydroxytryptamine (serotonin) receptor 2C0.39024Propiomazine
0.19362ADRA1A: alpha-1A adrenergic receptor
917NNNOlanzapine
OPRD1: opioid receptor, delta 10.40000Pimozide
0.15179ADRB2: beta-2 adrenergic receptor
918NNNBretylium tosylate
CXCR1: chemokine (C-X-C motif) receptor 10.44828Tolbutamide
0.094665ADRB2: beta-2 adrenergic receptor
919YNNCisapride
HTR1A: 5-hydroxytryptamine (serotonin) receptor 1A0.44444Metoclopramide
0.21367CHRM1: cholinergic receptor, muscarinic 1
922NYNBromocriptine
DRD1: dopamine receptor D10.26415Propiomazine
0.17500DRD2: dopamine receptor D2
923NNNOctreotide acetate
CCKAR: cholecystokinin A receptor0.34109Ceruletide
0.16860SSTR2
924NNNClozapine
NTSR2: neurotensin receptor 20.41026Levocabastine hydrochloride
0.10297HTR1B: 5-hydroxytryptamine (serotonin) receptor 1B
925NNNEpinephrine bitartrate
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.28125Pindolol
0.19131ADRB3: beta-3 adrenergic receptor
927NNNClozapine
OPRK1: opioid receptor, kappa 10.36667Dezocine
0.15982HTR4: 5-hydroxytryptamine (serotonin) receptor 4
928NNNGlyburide
HTR4: 5-hydroxytryptamine (serotonin) receptor 40.44516Cisapride
0.028484TBXA2R: thromboxane A2 receptor
929NNNTolterodine
ADRB1: beta-1 adrenergic receptor0.48387Dobutamine
0.16408CHRM1: cholinergic receptor, muscarinic 1
931NNNLevodopa
GPRC6A: G protein-coupled receptor, family C, group 6, member A0.31579Lysine hydrochloride
0.014484DRD2: dopamine receptor D2
932NNNConivaptan hydrochloride
HRH1: histamine receptor H10.37736Astemizole
0.053518AVPR2: arginine vasopressin receptor 2
933YYNRisperidone
ADRA2B: alpha-2B adrenergic receptor0.39474Clozapine
0.19075ADRA1A: alpha-1A adrenergic receptor
940NNNEletriptan hydrobromide
ADRB1: beta-1 adrenergic receptor0.45714Dobutamine hydrochloride
0.23627HTR1B: 5-hydroxytryptamine (serotonin) receptor 1B
941YNNZafirlukast
DRD2: dopamine receptor D20.42553Mesoridazine
0.094998LTB4R: leukotriene B4 receptor
942NNNBentiromide
AGTR1: angiotensin II receptor, type 10.39535Eprosartan
0.020002GRM8: glutamate receptor, metabotropic 8
944NNNVerapamil
ADRB3: beta-3 adrenergic receptor0.37500Dobutamine
0.23650ADRA1B: alpha-1B adrenergic receptor
945NNNSpiperone
HTR4: 5-hydroxytryptamine (serotonin) receptor 40.44444Clozapine
0.23774HTR7: 5-hydroxytryptamine (serotonin) receptor 7 (adenylate cyclase-coupled)
950NNNAminophylline
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.27660Risperidone
0.13353ADORA3: adenosine A3 receptor
951NNNOxymetazoline hydrochloride
CHRM2: cholinergic receptor, muscarinic 20.33333Tolterodine
0.16943ADRA2A: alpha-2A adrenergic receptor
952NNNNizatidine
HRH3: histamine receptor H30.32258Famotidine
0.12032HRH2: histamine receptor H2
954NNNAtropine
HRH3: histamine receptor H30.31250Maprotiline
0.24459CHRM1: cholinergic receptor, muscarinic 1
955NNNEpinephrine bitartrate
CXCR1: chemokine (C-X-C motif) receptor 10.21622Trimipramine
0.12052ADRA1A: alpha-1A adrenergic receptor
956NNNApafant
AGTR1: angiotensin II receptor, type 10.31250Irbesartan
0.20367PTAFR: platelet-activating factor receptor
957NYNCabergoline
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.47500Methysergide
0.18422DRD2: dopamine receptor D2
958NNYChlorpromazine hibenzate
HRH1: histamine receptor H10.42222Prochlorperazine
0.17178ADRA2A: alpha-2A adrenergic receptor
960NNNEpinastine hydrochloride
DRD5: dopamine receptor D50.48276Clozapine
0.23600HRH2: histamine receptor H2
961NNNAgomelatine
CHRM1: cholinergic receptor, muscarinic 10.46154Metoclopramide
0.13604HTR2C: 5-hydroxytryptamine (serotonin) receptor 2C
963NNNOlanzapine
MTNR1A: melatonin receptor 1A0.29032Agomelatine
0.14311ADRB3: beta-3 adrenergic receptor
966NNNCinnarizine
ADRA2B: alpha-2B adrenergic receptor0.42105Haloperidol
0.24263DRD2: dopamine receptor D2
968NNNAlfuzosin hydrochloride
HTR4: 5-hydroxytryptamine (serotonin) receptor 40.45238Cisapride
0.20748ADRA1A: alpha-1A adrenergic receptor
971NNNOctreotide acetate
LTB4R: leukotriene B4 receptor0.26316Zafirlukast
0.21466SSTR5: somatostatin receptor 5
973NNNCaffeine
CHRM1: cholinergic receptor, muscarinic 10.26087Pilocarpine
0.12335ADORA3: adenosine A3 receptor
975NNNCaffeine
HTR2C: 5-hydroxytryptamine (serotonin) receptor 2C0.28000Agomelatine
0.14048ADORA1: adenosine A1 receptor
976NNNVerapamil
DRD3: dopamine receptor D30.42105Chlorpromazine
0.23823ADRA2A: alpha-2A adrenergic receptor
977NNNIrbesartan
DRD2: dopamine receptor D20.41463Haloperidol
0.094658AGTR1: angiotensin II receptor, type 1
979NNNMethysergide
DRD3: dopamine receptor D30.35294Metoclopramide
0.18620HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A
982NNNCocaine
ADRA1A: alpha-1A adrenergic receptor0.38235Nifedipine
0.23539DRD1: dopamine receptor D1
984NNNAlprazolam
HTR2A: 5-hydroxytryptamine (serotonin) receptor 2A0.45161Clozapine
0.10700CXCR1: chemokine (C-X-C motif) receptor 1
989NNNDexmedetomidine
ADORA1: adenosine A1 receptor0.32000Theophylline sodium acetate
0.11754ADRA2A: alpha-2A adrenergic receptor
990NNNIrbesartan
ADRA1A: alpha-1A adrenergic receptor0.48780Spiperone
0.096750AGTR1: angiotensin II receptor, type 1
991NNNDobutamine hydrochloride
ADRA1A: alpha-1A adrenergic receptor0.48000Epinephrine hydrochloride
0.24577ADRB2: beta-2 adrenergic receptor
992NNNRenzapride
DRD2: dopamine receptor D20.44828Metoclopramide
0.16888HTR4: 5-hydroxytryptamine (serotonin) receptor 4
993NNNEpinephrine hydrochloride
CHRM1: cholinergic receptor, muscarinic 10.32143Profenamine hydrochloride
0.19188ADRA2A: alpha-2A adrenergic receptor
994NNNOxycodone
ADRA1A: alpha-1A adrenergic receptor0.32500Risperidone
0.14177OPRM1: opioid receptor, mu 1
995NNNPindolol
ADORA1: adenosine A1 receptor0.23333Ambuphylline
0.17450HTR4: 5-hydroxytryptamine (serotonin) receptor 4
996NNNBaclofen
ADRA2A: alpha-2A adrenergic receptor0.37037Epinephrine bitartrate
0.013422GABBR1: gamma-aminobutyric acid (GABA) B receptor, 1
998NNNSufentanil citrate
HRH1: histamine receptor H10.41667Doxylamine succinate
0.11037OPRM1: opioid receptor, mu 1
1000NNNMethoxamine hydrochloride
ADRA2C: alpha-2C adrenergic receptor0.42857Epinephrine hydrochloride
0.19685ADRA1B: alpha-1B adrenergic receptor